SCHEMBL19904686

SCHEMBL19904686

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCCC1)C1CCN(c2ccc3ccsc3c2)C1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.33
ALDH1A1 P00352 4/20 0.33
TSHR P16473 2/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTR1A P08908 2/20 0.33
UGCG Q16739 1/20 0.33
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SSTR3 P32745 2/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
SSTR1 P30872 1/20 0.31
NOTUM Q6P988 1/20 0.31
KDM4E B2RXH2 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904570 1.00 NAMPT (0.33) NAMPTALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL19904694 0.90 HTR1A (0.35) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904498 0.89 KDM4E (0.37) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904561 0.89 MCHR1 (0.36) HTR1AUGCG
SCHEMBL19904672 0.89 ALDH1A1 (0.38) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904363 0.89 ALDH1A1 (0.38) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904512 0.88 HTR1A (0.35) HTR1AUGCGSSTR3PDCD1CD274
SCHEMBL19904542 0.88 UGCG (0.40) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904389 0.88 UGCG (0.40) ALDH1A1TSHRHTTSMN1; SMN2HTR1A
SCHEMBL19904324 0.88 KDM4E (0.37) HTR1AUGCGSSTR3SSTR1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed