SCHEMBL19906119

SCHEMBL19906119

Cc1cc2nc(-c3ccc4cnccc4c3)sc2c(-c2ccc(Cl)cc2OC(C)(C)C)c1CC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.39
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CDC7 O00311 1/20 0.34
DBF4 Q9UBU7 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
INSR P06213 1/20 0.33
RET P07949 1/20 0.33
MET P08581 1/20 0.33
ROS1 P08922 1/20 0.33
PDGFRB P09619 1/20 0.33
FGFR1 P11362 1/20 0.33
SRC P12931 1/20 0.33
FGFR2 P21802 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905957 0.86 PTGDR2 (0.43) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906137 0.83 PTGDR2 (0.39) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906412 0.82 TP53 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905892 0.82 PTGDR2 (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905995 0.82 EIF4EBP1 (0.36) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906104 0.82 KDM4E (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906133 0.82 KMO (0.39) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906361 0.82 KDM4E (0.33) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906086 0.82 KDM4E (0.39) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906046 0.82 EIF4E (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed