SCHEMBL19906247

SCHEMBL19906247

Cc1cc2nc(-c3ccnc(-c4cnc5[nH]cc(C)c5c4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.40
BTK Q06187 8/20 0.37
ITK Q08881 8/20 0.37
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
SGK1 O00141 1/20 0.34
MAP3K12 Q12852 3/20 0.33
DYRK1A Q13627 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
AXL P30530 1/20 0.33
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906014 0.87 PTGDR2 (0.39) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906329 0.84 KDM4E (0.36) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19905852 0.84 KDM4E (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906265 0.84 KDM4E (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906236 0.83 PTGDR2 (0.38) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19905772 0.83 MAP4K4 (0.41) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL15333389 0.83 CYP3A4 (0.36) ABL1BTKITKCCNT1CCNA2
SCHEMBL15333762 0.83 CYP3A4 (0.36) ABL1BTKITKCCNT1CCNA2
SCHEMBL19906269 0.83 EIF4E (0.40) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906015 0.82 PIK3CG (0.38) KDM4EMEN1ALDH1A1KMT2APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed