SCHEMBL19936723

SCHEMBL19936723

Cc1[nH]cnc1CNc1ccc2nccnc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K8 P41279 1/20 0.45
ADRA2A P08913 2/20 0.43
ADRA2C P18825 2/20 0.43
KMT2A Q03164 6/20 0.39
WDR5 P61964 4/20 0.39
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 4/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
NFKB1 P19838 1/20 0.39
CYP2C19 P33261 1/20 0.39
KLK7 P49862 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
IP6K1 Q92551 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10883557 0.74 GAA (0.51) MAP3K8KMT2AWDR5KDM4EALDH1A1
SCHEMBL10882622 0.73 WDR5 (0.49) MAP3K8KMT2AWDR5SMN1; SMN2HRH2
SCHEMBL14035880 0.71 KDM4E (0.50) ADRA2AADRA2CKMT2AKDM4EALDH1A1
SCHEMBL10881527 0.68 HRH2 (0.43) MAP3K8ADRA2CKMT2AWDR5SMN1; SMN2
SCHEMBL14609411 0.67 ALDH1A1 (0.49) ADRA2AADRA2CKMT2AKDM4EALDH1A1
SCHEMBL11383611 0.67
SCHEMBL18669065 0.67 NPC1 (0.49) ADRA2AADRA2CKMT2AKDM4EALDH1A1
SCHEMBL10883114 0.66 MAP3K8 (0.43) MAP3K8ADRA2AADRA2CKMT2AWDR5
SCHEMBL10309415 0.65 ADRA2A (0.52) ADRA2AADRA2CKMT2AKDM4EALDH1A1
SCHEMBL10885778 0.65 TP53 (0.47) ADRA2CKMT2AWDR5ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802328-B1 TRYPTOLINE DERIVATIVES HAVING KINASE INHIBITORY ACTIVITY AND USES THEREOF X-CHEM INC (US) 2018-03-07 EP disclosed