SCHEMBL1994032

SCHEMBL1994032

CC(C)(C)OC(=O)N1CCC(NC(=O)c2ccc(N)nc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.56
USP30 Q70CQ3 3/20 0.53
SSTR5 P35346 2/20 0.52
PARP1 P09874 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
POLB P06746 1/20 0.50
EPHX1 P07099 1/20 0.50
GPR119 Q8TDV5 1/20 0.50
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
ALPL P05186 1/20 0.48
ALPI P09923 1/20 0.48
ALPG P10696 1/20 0.48
CA12 O43570 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2954898 0.87 HDAC4 (0.56) HDAC4USP30SSTR5L3MBTL1POLB
SCHEMBL12426680 0.86 HDAC4 (0.61) HDAC4USP30PARP1L3MBTL1POLB
SCHEMBL1994518 0.84 ALDH1A1 (0.45) HDAC4USP30L3MBTL1EPHX1GPR119
SCHEMBL2962009 0.84 HDAC4 (0.53) HDAC4USP30PARP1L3MBTL1POLB
SCHEMBL27861514 0.83 SSTR5 (0.52) SSTR5HDAC6
SCHEMBL28769906 0.83 HDAC4 (0.52) HDAC4USP30PARP1L3MBTL1POLB
SCHEMBL2952214 0.83 SSTR5 (0.55) HDAC4USP30SSTR5L3MBTL1POLB
SCHEMBL2951455 0.82 HPGDS (0.52) HDAC4USP30L3MBTL1POLBEPHX1
SCHEMBL2951452 0.81 L3MBTL1 (0.57) HDAC4USP30L3MBTL1POLBEPHX1
SCHEMBL29961114 0.81 HDAC4 (0.47) HDAC4USP30L3MBTL1GPR119HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2026-05-28 US disclosed
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2024-02-08 US disclosed
US-20210253578-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2021-08-19 US disclosed
US-20180155351-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2018-06-07 US disclosed
US-20170183352-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2017-06-29 US disclosed
US-9416136-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2016-08-16 US disclosed
US-8962630-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2015-02-24 US disclosed
EP-2331547-B1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2014-07-30 EP disclosed
US-20140135312-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2014-05-15 US disclosed
US-20130184285-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS (GB) 2013-07-18 US disclosed
US-8415355-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2013-04-09 US disclosed
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2011-06-23 US disclosed
EP-2331547-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS Novartis AG (CH) 2011-06-15 EP disclosed
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG 2010-04-29 US disclosed
WO-2010020675-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2010-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK9, CDK6, CDK7 HDAC4 722/4885USP30 3655/4885SSTR5 2403/4885
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20130184285-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20170183352-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20180155351-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20210253578-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885
US-20140135312-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 HDAC4 395/4885USP30 2946/4885SSTR5 3725/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.