SCHEMBL1994518

SCHEMBL1994518

CC(C)(C)OC(=O)N1CCC(NCC(=O)c2ccc(N)nc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
GPR119 Q8TDV5 8/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
USP30 Q70CQ3 1/20 0.43
ADORA2A P29274 1/20 0.43
HDAC4 P56524 1/20 0.42
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1994032 0.84 HDAC4 (0.56) ALDH1A1GPR119L3MBTL1MAPTKMT2A
SCHEMBL17961712 0.79 GPR119 (0.58) ALDH1A1GPR119L3MBTL1NPC1MAPT
SCHEMBL1990029 0.77 KMT2A (0.57) GPR119RAB9AKMT2AHDAC4
SCHEMBL1994519 0.77 USP30 (0.57) GPR119USP30
SCHEMBL19126445 0.76 TGFBR1 (0.51) ALDH1A1GPR119L3MBTL1NPC1MAPT
SCHEMBL3668808 0.76 LMNA (0.49) GPR119MAPTKMT2A
SCHEMBL29497122 0.75 DDB1 (0.60) GPR119MAPTKDM4EALOX5APFEN1
SCHEMBL611718 0.75 DDB1 (0.60) GPR119MAPTKDM4EALOX5APFEN1
SCHEMBL30490329 0.75 GPR119 (0.45) GPR119
SCHEMBL26641481 0.75 GPR119 (0.45) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2026-05-28 US disclosed
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2024-02-08 US disclosed
US-20210253578-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2021-08-19 US disclosed
US-20180155351-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2018-06-07 US disclosed
US-20170183352-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2017-06-29 US disclosed
US-9416136-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2016-08-16 US disclosed
US-8962630-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2015-02-24 US disclosed
EP-2331547-B1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2014-07-30 EP disclosed
US-20140135312-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2014-05-15 US disclosed
US-20130184285-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS (GB) 2013-07-18 US disclosed
US-8415355-B2 Pyrrolopyrimidine compounds and their uses NOVARTIS AG (CH) 2013-04-09 US disclosed
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2011-06-23 US disclosed
EP-2331547-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS Novartis AG (CH) 2011-06-15 EP disclosed
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG 2010-04-29 US disclosed
WO-2010020675-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2010-02-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK9, CDK6, CDK7 ALDH1A1 3935/4885GPR119 3309/4885L3MBTL1 1901/4885
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20130184285-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20170183352-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20180155351-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20210253578-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885
US-20140135312-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 ALDH1A1 3688/4885GPR119 3780/4885L3MBTL1 1362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.