SCHEMBL19944650

SCHEMBL19944650

CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)N[C@H](/C=C(\Cl)S(C)(=O)=O)CC(=O)O

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.66
CASP7 P55210 2/20 0.66
CASP9 P55211 2/20 0.66
CASP10 Q92851 1/20 0.66
CASP1 P29466 2/20 0.59
CTSL P07711 9/20 0.58
CTSB P07858 6/20 0.58
PSMB5 P28074 3/20 0.56
CTSK P43235 3/20 0.56
PSMB1 P20618 1/20 0.54
PSMB2 P49721 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15462664 0.87 CASP3 (0.73) CASP3CASP7CASP9CASP10CASP1
SCHEMBL19944919 0.86 CASP3 (0.70) CASP3CASP7CASP9CASP1CTSL
SCHEMBL15462725 0.83 CASP3 (0.78) CASP3CASP7CASP9CASP10CASP1
SCHEMBL15462693 0.83 CASP3 (0.78) CASP3CASP7CASP9CASP10CASP1
SCHEMBL20356006 0.83 CASP3 (0.78) CASP3CASP7CASP9CASP10CASP1
SCHEMBL4427171 0.82 PSMB1 (0.71) CTSLCTSBPSMB5CTSKPSMB1
SCHEMBL27543993 0.82 PSMB1 (0.71) CTSLCTSBPSMB5CTSKPSMB1
SCHEMBL9962302 0.80 CASP3 (0.81) CASP3CASP7CASP9CASP10CASP1
SCHEMBL19944654 0.80 CASP1 (0.66) CASP3CASP7CASP9CASP10CASP1
SCHEMBL16376143 0.80 CASP3 (0.58) CASP3CASP7CASP9CASP10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697246-B1 SELECTIVE CYSTEINE PROTEASE INHIBITORS AND USES THEREOF GENESIS TECH LIMITED (BB) 2018-03-07 EP disclosed