SCHEMBL19944654

SCHEMBL19944654

CCOC(=O)/C=C/[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.66
CASP3 P42574 1/20 0.66
CASP4 P49662 1/20 0.66
CASP7 P55210 1/20 0.66
CASP9 P55211 1/20 0.66
CASP8 Q14790 1/20 0.66
CASP10 Q92851 1/20 0.66
CTSL P07711 13/20 0.65
CTSB P07858 7/20 0.58
CTSK P43235 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15462666 0.87 CASP3 (0.73) CASP1CASP3CASP4CASP7CASP9
SCHEMBL19944919 0.85 CASP3 (0.70) CASP1CASP3CASP4CASP7CASP9
SCHEMBL19944665 0.84 CASP3 (0.61) CASP1CASP3CASP4CASP7CASP9
SCHEMBL27543993 0.82 PSMB1 (0.71) CTSLCTSBCTSK
SCHEMBL4427171 0.82 PSMB1 (0.71) CTSLCTSBCTSK
SCHEMBL19944562 0.81 CTSL (0.54) CASP1CASP3CASP4CASP7CASP9
SCHEMBL7612532 0.80 CTSK (0.71) CTSLCTSBCTSK
SCHEMBL7612544 0.80 CTSK (0.71) CTSLCTSBCTSK
SCHEMBL19944650 0.80 CASP3 (0.66) CASP1CASP3CASP7CASP9CASP10
SCHEMBL30070594 0.80 CTSL (0.76) CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697246-B1 SELECTIVE CYSTEINE PROTEASE INHIBITORS AND USES THEREOF GENESIS TECH LIMITED (BB) 2018-03-07 EP disclosed