SCHEMBL19944665

SCHEMBL19944665

CCOC(=O)/C=C/[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)CNC(=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 8/20 0.61
CASP7 P55210 5/20 0.61
CASP1 P29466 4/20 0.61
CASP9 P55211 2/20 0.61
CASP4 P49662 2/20 0.61
CASP8 Q14790 1/20 0.61
CASP10 Q92851 1/20 0.61
CTSL P07711 6/20 0.51
LGMN Q99538 1/20 0.47
CTSB P07858 2/20 0.46
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20052410 0.91 CASP3 (0.58) CASP3CASP7CASP1CASP9CASP4
SCHEMBL19944785 0.91 CASP3 (0.58) CASP3CASP7CASP1CASP9CASP4
SCHEMBL15462666 0.85 CASP3 (0.73) CASP3CASP7CASP1CASP9CASP4
SCHEMBL19944654 0.84 CASP1 (0.66) CASP3CASP7CASP1CASP9CASP4
SCHEMBL18782028 0.80 CASP3 (0.77) CASP3CASP7CASP1CASP9CASP4
SCHEMBL11112981 0.80 CYP3A4 (0.53) CTSLCTSBMAPK1
SCHEMBL29434574 0.78 CTSB (0.62) CTSLCTSBMAPK1
SCHEMBL29434511 0.77 CTSB (0.56) CTSLCTSB
SCHEMBL15462686 0.76 CASP3 (1.00) CASP3CASP7CASP1CASP9CASP4
SCHEMBL29544585 0.76 REN (0.54) CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697246-B1 SELECTIVE CYSTEINE PROTEASE INHIBITORS AND USES THEREOF GENESIS TECH LIMITED (BB) 2018-03-07 EP disclosed