SCHEMBL1994560

SCHEMBL1994560

O=C(Cl)c1ccc(N2C(=O)c3ccc(C(=O)Cl)cc3C2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 11/20 0.57
CA1 P00915 8/20 0.57
CA12 O43570 6/20 0.57
CA2 P00918 5/20 0.56
CA4 P22748 3/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
GFER P55789 1/20 0.55
ESR1 P03372 2/20 0.54
ESR2 Q92731 2/20 0.54
NPSR1 Q6W5P4 2/20 0.54
SCN2A Q99250 1/20 0.53
ALDH1A1 P00352 2/20 0.50
MAPT P10636 1/20 0.49
POLB P06746 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1618166 0.90 ESR1 (0.61) CA9CA1CA12CA2CA4
SCHEMBL1995596 0.85 S100B (0.57) MEN1KMT2AESR1NPSR1ALDH1A1
SCHEMBL17281691 0.84 PTGES (0.61) CA9CA1CA12CA2CA4
SCHEMBL9339007 0.82 CA9 (0.77) CA9CA1CA12CA2CA4
SCHEMBL4234750 0.81 CA9 (0.77) CA9CA1CA12CA2CA4
SCHEMBL15081236 0.80 CA9 (0.51) CA9CA1CA12CA2CA4
SCHEMBL15176768 0.80 MAP4K4 (0.45) CA9CA1CA12CA2CA4
SCHEMBL27464004 0.80 POLB (0.47) CA9CA1CA2CA4MEN1
SCHEMBL17946636 0.80 MEN1 (0.59) CA9CA1CA12CA2CA4
SCHEMBL14016924 0.79 CA9 (0.64) CA9CA1CA12CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2338485-A1 Substituted 1,3-dioxoisoindolines as medicine Grünenthal GmbH (DE) 2011-06-29 EP disclosed
US-5162489-A Containing a 1,1,3-trimethylphenylindane moiety AKZO N.V. (NL) 1992-11-10 US disclosed
US-4980504-A WHICH HAVE HIGH GLASS TRANSITION TEMPERATURES AKZO N.V. (NL) 1990-12-25 US disclosed
EP-0357106-A1 Aromatic amide groups-containing diamines and polymers prepared therefrom AKZO N.V. (NL) 1990-03-07 EP disclosed