SCHEMBL19953055

SCHEMBL19953055

Fc1cc(Cl)ccc1-n1cnc(Cl)c1-c1c(F)cccc1F

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.37
PTGS1 P23219 1/20 0.37
FGFR1 P11362 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
TRPM5 Q9NZQ8 1/20 0.35
PDE2A O00408 1/20 0.34
PDE10A Q9Y233 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953173 0.82 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL19952995 0.81 HCAR1 (0.40) PTGS2PTGS1GABRG2GABRB3GABRA5
SCHEMBL19953169 0.75 CYP3A4 (0.43) EGLN2TRPM5PDE2APDE10A
SCHEMBL1073380 0.72 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL19953095 0.68 PDE4B (0.38) EGLN2TRPM5PDE2APDE10A
SCHEMBL19953199 0.68 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL19953048 0.68 PTGS2 (0.42) PTGS2PTGS1GABRG2GABRB3GABRA5
SCHEMBL1074163 0.68 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL15638551 0.66 MAP3K14 (0.42) FGFR1
SCHEMBL1074104 0.66 PTGS2 (0.47) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed