SCHEMBL19953586

SCHEMBL19953586

CCOC(=O)C1c2ccccc2CC(=O)N1C.CCOC(=O)Cc1ccccc1C(Br)C(=O)OCC

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.35
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NOTUM Q6P988 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
LMNA P02545 1/20 0.33
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
GRM7 Q14831 1/20 0.32
TBXAS1 P24557 1/20 0.32
NAMPT P43490 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953669 0.82 MEN1 (0.42) ALDH1A1KDM4ENOTUMLMNAAPOBEC3A
SCHEMBL19953657 0.78 PKM (0.47) ALDH1A1CYP4F2CYP4A11TBXAS1
SCHEMBL19960636 0.69 HDAC4 (0.43) NOTUMGRM7
SCHEMBL20166097 0.67 GRM7 (0.39) ALDH1A1KDM4ENOTUMLMNAGRM7
SCHEMBL19960628 0.67 PKM (0.48) ALDH1A1CYP4F2CYP4A11TBXAS1
SCHEMBL20113096 0.67 GRM7 (0.55) ALDH1A1KDM4EGRM7MAPT
SCHEMBL4028087 0.66 TSHR (0.49) ALDH1A1KDM4ECYP4F2CYP4A11LMNA
SCHEMBL19953652 0.65 ACE (0.47) ACENOTUMGRM7
SCHEMBL11273360 0.65 PIN1 (0.41) CYP4F2CYP4A11LMNA
SCHEMBL19953522 0.65 ACE (0.47) ACENOTUMGRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed