SCHEMBL199603

SCHEMBL199603

N#CC[CH]c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
CYP2A6 P11509 1/20 0.42
MAOB P27338 3/20 0.39
MAOA P21397 2/20 0.39
TSHR P16473 2/20 0.36
IDO1 P14902 2/20 0.35
PAM P19021 1/20 0.35
HTT P42858 1/20 0.35
MCL1 Q07820 1/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6599473 0.87 TP53 (0.38) ALDH1A1LMNA
SCHEMBL3012608 0.78 MAOB (0.49) MAOBMAOAIDO1PAML3MBTL1
SCHEMBL1002069 0.78 MAOB (0.49) MAOBMAOAIDO1PAML3MBTL1
SCHEMBL3240426 0.76 ALDH1A1 (0.39) ALDH1A1CYP2A6MAOBMAOATSHR
SCHEMBL8110092 0.75 ALDH1A1 (0.42) ALDH1A1CYP2A6MAOBMAOATSHR
SCHEMBL6258270 0.75 ALDH1A1 (0.42) ALDH1A1CYP2A6MAOBMAOATSHR
SCHEMBL16957356 0.74 NFE2L2 (0.52) NPC1RAB9A
SCHEMBL16956466 0.74 CHRM5 (0.47) ALDH1A1MAOBGAA
SCHEMBL1162641 0.73 MAOA (0.36) ALDH1A1CYP2A6MAOBMAOAL3MBTL1
Styrene SCHEMBL28107406 0.73 ALDH1A1 (0.58) ALDH1A1MAOBMAOATSHRIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 232 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023214119-A1 AZETIDINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, PREPARATION METHODS AND THEIR USES IN THE TREATMENT OF CNS DISORDERS EQUINORM LTD (FI) 2023-11-09 WO claimed
US-20070287699-A1 ANTIVIRAL AGENTS VIROBAY, INC. (US) 2007-12-13 US claimed
WO-2007130499-A2 ANTIVIRAL AGENTS VIROBAY, INC. (US) 2007-11-15 WO claimed
EP-1594835-A4 METHOD OF PREPARATION OF HETEROCYCLIC MOLECULES WITH PHARMACEUTICAL PHARMACEUTICAL EXCIPIENT COSMECEUTICAL AGROCHEMICAL AND INDUSTRIAL USES AUSPEX PHARMACEUTICALS INC (US) 2007-05-02 EP claimed
US-20060173199-A1 Method of preparation of heterocyclic molecules with pharmaceutical, pharmaceutical excipient, cosmeceutical, agrochemical and industrial uses HONG BORCHERNG 2006-08-03 US claimed
EP-1594835-A2 METHOD OF PREPARATION OF HETEROCYCLIC MOLECULES WITH PHARMACEUTICAL PHARMACEUTICAL EXCIPIENT COSMECEUTICAL AGROCHEMICAL AND INDUSTRIAL USES Auspex Pharmaceuticals, Inc. (US) 2005-11-16 EP claimed
WO-2004064745-A2 METHOD OF PREPARATION OF HETEROCYCLIC MOLECULES WITH PHARMACEUTICAL PHARMACEUTICAL EXCIPIENT COSMECEUTICAL AGROCHEMICAL AND INDUSTRIAL USES AUSPEX PHARMACEUTICALS, INC. (US) 2004-08-05 WO claimed
EP-0477646-B1 Substituted 5-alkoxy-1,2,4-triazol-3-(thi)ones BAYER AG (DE) 1995-03-01 EP claimed
EP-0283876-B1 Substituted triazolinones BAYER AG (DE) 1994-07-20 EP claimed
EP-0294666-B1 Substituted triazolinones BAYER AG (DE) 1994-02-16 EP claimed
US-5276008-A Herbicides and plant growth regulators BAYER AKTIENGESELLSCHAFT (DE) 1994-01-04 US claimed
EP-0332991-B1 Substituted triazoles BAYER AG (DE) 1993-11-10 EP claimed
EP-0398096-B1 SUBSTITUTED TRIAZOLONES BAYER AG (DE) 1993-10-13 EP claimed
EP-0412358-B1 3-AMINO-5-AMINOCARBONYL-1,2,4-TRIAZOLE DERIVATIVES BAYER AG (DE) 1993-09-29 EP claimed
EP-0415196-B1 SUBSTITUTED 4,5-DIAMINO-1,2,4-TRIAZOL-3-(THI)ONES BAYER AG (DE) 1993-03-24 EP claimed
EP-0399285-B1 PROCESS FOR THE PREPARATION OF 3-AMINO-5-AMINOCARBONYL-1,2,4-TRIAZOLE DERIVATIVES BAYER AG (DE) 1992-09-30 EP claimed
US-5082490-A HERBICIDAL SUBSTITUTED 4,5-DIAMINO-1,2,4-TRIAZOL-3-(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 1992-01-21 US claimed
US-5061311-A SUBSTITUTED TRIAZOLINONE HERBICIDES AND PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1991-10-29 US claimed
EP-0298371-B1 SUBSTITUTED TRIAZOLINONES BAYER AG (DE) 1991-10-02 EP claimed
US-5051517-A Reacting a chloroformidine hydrochloride with an oxamohydrazide, forming bonds between carbon and nitrogen and cyclization BAYER AKTIENGESELLSCHAFT (DE) 1991-09-24 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070287699-A1 ANTIVIRAL AGENTS EIF2AK2, MAVS, ZC3HAV1 ALDH1A1 1759/4885CYP2A6 2507/4885MAOB 3428/4885
US-20060173199-A1 Method of preparation of heterocyclic molecules with pharmaceutical, pharmaceutical excipient, cosmeceutical, agrochemical and industrial uses LSS, DHPS, CYP51A1 ALDH1A1 1435/4885CYP2A6 51/4885MAOB 232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.