SCHEMBL19962013

SCHEMBL19962013

CN(C(=O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)c1c(F)c(F)c(F)c(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)C(=O)N(C)c2ccc3scnc3c2)c1F)c1ccc2sccc2c1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.34
PIN1 Q13526 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18180150 0.93 TAS1R3 (0.34) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL18179993 0.93 TAS1R3 (0.34) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL19962038 0.91 PIN1 (0.39) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL19962065 0.89 NOS2 (0.33) PYGLPDE10A
SCHEMBL19962046 0.88 BACE1 (0.34) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL19962042 0.88 PYGL (0.34) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL19962064 0.88 PIN1 (0.36) PYGLPIN1TAS1R3TAS1R1PDE10A
SCHEMBL19969001 0.87 TAS1R3 (0.31) PYGLTAS1R3TAS1R1
SCHEMBL19962014 0.87 PYGL (0.36) PYGLPIN1PDE10A
SCHEMBL19962010 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180072997-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY 2018-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180072997-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION EIF2AK2, POLR2H, POLR2E PYGL 498/4885PIN1 1030/4885TAS1R3 4630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.