SCHEMBL19965160

SCHEMBL19965160

Clc1cccc(Oc2cccc(N3Cc4ccccc4S3)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAP4K4 O95819 1/20 0.40
FFAR4 Q5NUL3 2/20 0.34
BCHE P06276 1/20 0.34
DCK P27707 1/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
SLC6A2 P23975 3/20 0.32
SLC6A4 P31645 3/20 0.32
SLC6A3 Q01959 3/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
HTR1A P08908 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19965080 0.81 LMNA (0.38) MAP4K4FFAR4LMNAPIM1PIM2
SCHEMBL19965054 0.74 MAP3K5 (0.47) CYP1A2CYP2C9CYP2C19MAP4K4PIM1
SCHEMBL19965064 0.74 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19MAP4K4FFAR4
SCHEMBL21124601 0.73 FFAR4 (0.60) CYP1A2CYP2C9CYP2C19MAP4K4FFAR4
SCHEMBL30918019 0.71 CASP6 (0.42) CYP1A2CYP2C9CYP2C19MAPTLMNA
SCHEMBL19965171 0.70 BRAF (0.36) MAP4K4FFAR4LMNAHRH3GRM5
SCHEMBL6791132 0.69 HTR3A (0.55) CYP1A2CYP2C9CYP2C19MAP4K4DCK
SCHEMBL8115420 0.68 MAP4K4 (0.59) CYP1A2CYP2C9CYP2C19MAP4K4SCN5A
SCHEMBL959384 0.68 L3MBTL1 (0.57) CYP1A2CYP2C9CYP2C19MAP4K4PIM1
SCHEMBL19965170 0.65 KDM4E (0.39) CYP1A2CYP2C9CYP2C19HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049324-A1 MONOCYCLIC COMPOUNDS USEFUL AS GPR120 MODULATORS NUMERATE, INC. (US) 2018-03-15 WO disclosed