SCHEMBL19970087

SCHEMBL19970087

Cc1ccccc1-c1nc(NSc2cccc(NC3CCC(C(=O)O)C3)n2)ccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 3/20 0.35
SYK P43405 2/20 0.34
DYRK3 O43781 1/20 0.33
MAP4K4 O95819 1/20 0.33
ERBB2 P04626 1/20 0.33
PIM1 P11309 1/20 0.33
MARK3 P27448 1/20 0.33
PLK1 P53350 1/20 0.33
CAMK2B Q13554 1/20 0.33
CDC42BPA Q5VT25 1/20 0.33
PIM3 Q86V86 1/20 0.33
MINK1 Q8N4C8 1/20 0.33
SRPK1 Q96SB4 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
MAP3K20 Q9NYL2 1/20 0.33
MAP4K5 Q9Y4K4 1/20 0.33
MAPK3 P27361 1/20 0.33
VCP P55072 1/20 0.32
NUDT1 P36639 1/20 0.31
IL1B P01584 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770784 0.96 SYK (0.38) CCNT1SYKVCPNUDT1IL1B
SCHEMBL19970019 0.95 MAPK3 (0.38) CCNT1SYKMAPK3NUDT1IL1B
SCHEMBL19970021 0.95 MAPK3 (0.38) CCNT1SYKMAPK3NUDT1IL1B
SCHEMBL19970024 0.95 MAPK3 (0.38) CCNT1SYKMAPK3NUDT1IL1B
SCHEMBL23770790 0.86 IL1B (0.32) CCNT1IL1BCCNKCCNE1CDK2
SCHEMBL23770573 0.86 CCNT1 (0.36) CCNT1PIM1IL1BMEN1CYP1A2
SCHEMBL23770848 0.86 IL1B (0.33) IL1BCTSA
SCHEMBL23770706 0.85 SMN1; SMN2 (0.36) CCNT1PIM1MEN1TSHRKMT2A
SCHEMBL19951335 0.85 SYK (0.42) SYKVCPNUDT1IL1BEPHX2
SCHEMBL19951403 0.84 MAPK3 (0.44) CCNT1DYRK3MAP4K4ERBB2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11066369-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease NOVARTIS AG (CH) 2021-07-20 US disclosed
US-10450273-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease NOVARTIS AG (CH) 2019-10-22 US disclosed
US-20180072673-A1 N-(pyridin-2-yl)pyridine-sulfonamide Derivatives and their Use in the Treatment of Disease NOVARTIS AG (CH) 2018-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11066369-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease CFTR, P2RY1, P2RX5 CCNT1 4170/4885SYK 689/4885DYRK3 2450/4885
US-20180072673-A1 N-(pyridin-2-yl)pyridine-sulfonamide Derivatives and their Use in the Treatment of Disease CFTR, P2RY1, P2RX5 CCNT1 4170/4885SYK 689/4885DYRK3 2450/4885
US-10450273-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease CFTR, P2RY1, P2RX5 CCNT1 4170/4885SYK 689/4885DYRK3 2450/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.