SCHEMBL19970150

SCHEMBL19970150

CC(C)(C)OC(=O)NC1=CC=CC(S)N1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 4/20 0.36
NFKB2 Q00653 4/20 0.36
RELA Q04206 4/20 0.36
BRD4 O60885 2/20 0.34
CREBBP Q92793 2/20 0.34
GAA P10253 1/20 0.32
CYP17A1 P05093 1/20 0.32
ATR Q13535 1/20 0.32
EPHX2 P34913 1/20 0.32
PTPN11 Q06124 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29415863 0.71 CYP17A1 (0.37) GAACYP17A1ATRPTPN11CA1
SCHEMBL20689331 0.63 GAA (0.35) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL13055402 0.62 CYP17A1 (0.59) GAACYP17A1PTPN11CA1
SCHEMBL21155495 0.62 GAA (0.35) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL29032266 0.62 NFKB1 (0.39) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL14110260 0.62 EPHX2 (0.42) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL977487 0.60 CYP17A1 (0.54) CYP17A1PTPN11CA1
SCHEMBL28269645 0.59 NFKB1 (0.42) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL27991298 0.59 NFKB1 (0.42) NFKB1NFKB2RELAGAACYP17A1
SCHEMBL2880191 0.59 LMNA (0.54) BRD4GAACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10450273-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease NOVARTIS AG (CH) 2019-10-22 US disclosed
US-20180072673-A1 N-(pyridin-2-yl)pyridine-sulfonamide Derivatives and their Use in the Treatment of Disease NOVARTIS AG (CH) 2018-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180072673-A1 N-(pyridin-2-yl)pyridine-sulfonamide Derivatives and their Use in the Treatment of Disease CFTR, P2RY1, P2RX5 NFKB1 1236/4885NFKB2 1404/4885RELA 1082/4885
US-10450273-B2 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease CFTR, P2RY1, P2RX5 NFKB1 1236/4885NFKB2 1404/4885RELA 1082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.