SCHEMBL19976782

SCHEMBL19976782

CCOCCN/C(=N/C(=O)c1ccc(F)c(F)c1)Nc1n[nH]c2c(C(F)(F)F)cccc12

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.36
TRPA1 O75762 2/20 0.35
EGFR P00533 1/20 0.34
HDAC6 Q9UBN7 3/20 0.33
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
GSK3B P49841 2/20 0.32
KDR P35968 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
FGFR1 P11362 2/20 0.32
FGFR2 P21802 2/20 0.32
FGFR3 P22607 2/20 0.32
ABL1 P00519 1/20 0.32
BCR P11274 1/20 0.32
KDM4E B2RXH2 1/20 0.32
FGFR4 P22455 1/20 0.32
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976768 0.91 MAPK1 (0.38) MAPK1TRPA1EGFRHDAC6GSK3B
SCHEMBL19976805 0.86 ALDH1A1 (0.36) MAPK1TRPA1GSK3BHPGDTSHR
SCHEMBL19976781 0.85 TRPA1 (0.35) MAPK1TRPA1EGFRABL1BCR
SCHEMBL19976731 0.85 MAPK1 (0.42) MAPK1HDAC6GSK3BFGFR1FGFR2
SCHEMBL19976812 0.84 GSK3B (0.51) MAPK1TRPA1HDAC6GSK3BFGFR1
SCHEMBL19976804 0.83 TRPA1 (0.37) TRPA1EGFRHDAC6GSK3BKDR
SCHEMBL19976815 0.83 GSK3B (0.44) MAPK1TRPA1HDAC6GSK3B
SCHEMBL19976858 0.82 MAPK1 (0.46) MAPK1HDAC6GSK3BFGFR1FGFR2
SCHEMBL19976764 0.81 GSK3B (0.48) MAPK1TRPA1HDAC6GSK3BFGFR1
SCHEMBL19976828 0.80 GSK3B (0.49) MAPK1TRPA1HDAC6GSK3BFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9920012-B2 Indazole guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2018-03-20 US disclosed