SCHEMBL19977054

SCHEMBL19977054

CC(NC(=O)c1cccs1)C(=O)Nc1ccccc1N1CCNCC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.57
NPSR1 Q6W5P4 3/20 0.57
LMNA P02545 3/20 0.57
TSHR P16473 2/20 0.57
MAPK1 P28482 1/20 0.57
ALDH1A1 P00352 6/20 0.54
GAA P10253 1/20 0.53
HTT P42858 2/20 0.52
CHEK1 O14757 11/20 0.52
ALOX12 P18054 2/20 0.51
KMT2A Q03164 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MEN1 O00255 1/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19977040 0.90 MAPT (0.71) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL19976917 0.88 ALDH1A1 (0.66) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL19976936 0.87 SRPK1 (0.48) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL16993927 0.84 HSPA1A (0.55) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL19977049 0.84 ALDH1A1 (0.55) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL16993938 0.82 MAPT (0.52) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL19976964 0.81 L3MBTL1 (0.58) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL19977129 0.80 ALDH1A1 (0.57) MAPTNPSR1LMNATSHRMAPK1
SCHEMBL5558994 0.78 POLB (0.66) MAPTNPSR1TSHRMAPK1ALDH1A1
SCHEMBL19976901 0.77 GAA (0.59) MAPTNPSR1LMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed