SCHEMBL19980338

SCHEMBL19980338

CC(C)(C)OC(=O)NCC1COc2ccccc2NC1=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 10/20 0.43
IDO1 P14902 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
EPHX2 P34913 1/20 0.41
GAA P10253 1/20 0.40
MAPK10 P53779 1/20 0.40
TSHR P16473 1/20 0.39
PARP1 P09874 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22048691 0.89 ACACB (0.42) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL21156303 0.82 GAA (0.35) IDO1KDM4EALDH1A1HPGDEPHX2
SCHEMBL3485743 0.81 GAA (0.57) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL1561667 0.81 GAA (0.57) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL1561665 0.81 GAA (0.57) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL31213772 0.75 DRD2 (0.41) IDO1KDM4EALDH1A1HPGDEPHX2
SCHEMBL29960414 0.74 IDO1 (0.48) IDO1ALDH1A1EPHX2MAPK10PARP1
SCHEMBL18368150 0.74 RIPK1 (0.52) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL21156863 0.74 RIPK1 (0.52) RIPK1IDO1EPHX2GAAMAPK10
SCHEMBL31544619 0.74 MTNR1A (0.67) ALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2956452-B1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2018-03-21 EP disclosed