SCHEMBL19982244

SCHEMBL19982244

CC(Cc1ccc(OCc2ccccc2)cc1)NC(=O)CN1CCN(C(=O)C2CCCN2C)CC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
RAB9A P51151 2/20 0.48
ACE P12821 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TP53 P04637 1/20 0.46
CACNA1B Q00975 1/20 0.45
YAP1 P46937 4/20 0.45
CHRNB2 P17787 1/20 0.44
CHRNA5 P30532 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNA4 P43681 1/20 0.44
LTA4H P09960 1/20 0.44
EPHX2 P34913 1/20 0.44
LMNA P02545 4/20 0.44
HTT P42858 2/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.43
SLC2A1 P11166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982261 0.91 LMNA (0.51) ALDH1A1RAB9AACELMNAHTT
SCHEMBL22929113 0.81 ACE (0.46) ALDH1A1RAB9AACESMN1; SMN2TP53
SCHEMBL19982125 0.80 YAP1 (0.57) ACEYAP1GAA
SCHEMBL19982079 0.78 YAP1 (0.73) YAP1GAA
SCHEMBL19975033 0.73 YAP1 (0.62) ALDH1A1RAB9AYAP1LMNAGAA
SCHEMBL19975035 0.73 YAP1 (0.62) ALDH1A1RAB9AYAP1LMNAGAA
SCHEMBL20111166 0.72 HDAC1 (0.61) ALDH1A1SMN1; SMN2CHRNB2CHRNA5CHRNA7
SCHEMBL8189803 0.72 KMT2A (0.58) ALDH1A1SMN1; SMN2LMNAMAPTKDM4E
SCHEMBL22929115 0.71 ITGB1 (0.46) ALDH1A1ACELTA4HKDM4E
SCHEMBL1302762 0.71 SMN1; SMN2 (0.57) ALDH1A1RAB9ASMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053446-A1 YAP1 INHIBITORS THAT TARGET THE INTERACTION OF YAP1 WITH OCT4 H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2018-03-22 WO disclosed