SCHEMBL19983031

SCHEMBL19983031

CC(C)(C)OC(=O)NOCCOc1c(F)cccc1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.40
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
CA12 O43570 6/20 0.37
CA1 P00915 6/20 0.37
CA2 P00918 5/20 0.37
CA9 Q16790 5/20 0.37
KMT2A Q03164 1/20 0.35
AAK1 Q2M2I8 2/20 0.35
PTPN1 P18031 1/20 0.35
CA7 P43166 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ATM Q13315 1/20 0.34
SYK P43405 1/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983074 0.79 KMT2A (0.40) SCN9ACTSSCTSKCA12CA1
SCHEMBL32665252 0.77 CHRNB2 (0.48) CA12CA1CA2CA9
SCHEMBL19983027 0.76 LMNA (0.41) SCN9ACTSSCTSKKMT2ARAB9A
SCHEMBL32665418 0.74 CA12 (0.50) CTSSCTSKCA12CA1CA2
SCHEMBL18921519 0.74 CTSS (0.39) SCN9ACTSSCTSKCA12CA1
SCHEMBL21601400 0.74 SCN9A (0.51) SCN9ACA12CA1CA2CA9
SCHEMBL12671642 0.73 KCNA5 (0.41) SCN9ACTSSCTSKCA12CA1
SCHEMBL1549969 0.72 ALDH1A1 (0.46) SCN9ACTSSCTSKCA12CA1
SCHEMBL32665511 0.72 CA12 (0.51) CA12CA1CA2CA9KMT2A
SCHEMBL32665495 0.72 NPC1 (0.51) KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed