SCHEMBL19983438

SCHEMBL19983438

Fc1cnc(N2CCN(S)CC2)nc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.46
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
DRD2 P14416 1/20 0.43
HTR1A P08908 2/20 0.42
OGA O60502 1/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24126297 0.80 SIGMAR1 (0.46) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL20182980 0.78 SIGMAR1 (0.46) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL18248348 0.77 SIGMAR1 (0.44) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL18248327 0.77 SIGMAR1 (0.44) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL30775408 0.75 KDM4E (0.61) SIGMAR1KDM4E
SCHEMBL2274356 0.75 ALDH1A1 (0.59) SIGMAR1KDM4ECYP1A2CYP2C9HTR1A
SCHEMBL28612099 0.75 HTR1A (0.46) SIGMAR1KDM4ECYP1A2GAACYP2C9
Hydrochloric Acid SCHEMBL25310447 0.73 ALDH1A1 (0.62) SIGMAR1KDM4ECYP1A2CYP2C9HTR1A
SCHEMBL18248260 0.73 SIGMAR1 (0.42) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL5368547 0.73 L3MBTL1 (0.49) SIGMAR1KDM4ECYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053126-A1 INHIBITION OF BMP SIGNALING, COMPOUNDS, COMPOSITIONS AND USES THEREOF VANDERBILT UNIVERSITY (US) 2018-03-22 WO disclosed