SCHEMBL19984374

SCHEMBL19984374

CNc1cc(OC2CC2)cc(F)c1N

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 6/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
KAT6A Q92794 1/20 0.32
HRH3 Q9Y5N1 1/20 0.31
EPHX2 P34913 1/20 0.30
DGAT1 O75907 1/20 0.30
SOAT1 P35610 1/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18519062 0.82 PTGS1 (0.36) ACACBPTGS1PTGS2KAT6AEPHX2
SCHEMBL18471239 0.71 PTGS1 (0.40) ACACBPTGS1PTGS2KAT6AHRH3
SCHEMBL107465 0.69 ALDH1A1 (0.34) FEN1
SCHEMBL20444243 0.67 ALDH1A1 (0.42) ACACBEPHX2PTPN1
SCHEMBL15045862 0.67 KDM1A (0.39) ACACBPTGS1PTGS2KAT6AEPHX2
SCHEMBL31508140 0.67 ALDH1A1 (0.43) ACACBPTGS1PTGS2HRH3EPHX2
SCHEMBL22470625 0.67 HTR2A (0.33)
SCHEMBL20600826 0.66 HDAC1 (0.34)
SCHEMBL30525820 0.66 HDAC1 (0.34)
SCHEMBL17949374 0.65 PGR (0.38) ACACBPTGS1PTGS2KAT6AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3279187-B1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO (JP) 2021-06-02 EP disclosed
US-20190144396-A1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO., LTD. (JP) 2019-05-16 US disclosed
US-10233156-B2 9-membered fused ring derivative SHIONOGI & CO., LTD. (JP) 2019-03-19 US disclosed
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO., LTD. (JP) 2018-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE ACSS2, AGTR2, ACSL3 ACACB 7/4885PTGS1 3793/4885PTGS2 2320/4885
US-20190144396-A1 9-MEMBERED FUSED RING DERIVATIVE ACSS2, AGTR2, ACSL3 ACACB 7/4885PTGS1 3793/4885PTGS2 2320/4885
US-10233156-B2 9-membered fused ring derivative AGTR2, ACSS2, ACSL3 ACACB 5/4885PTGS1 3917/4885PTGS2 2224/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.