SCHEMBL19984536

SCHEMBL19984536

COC(=O)C1CCCN1Sc1ccc(Br)cc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
HPGD P15428 2/20 0.43
MAPK1 P28482 2/20 0.42
MAPT P10636 6/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
ITGB2 P05107 2/20 0.38
ICAM1 P05362 2/20 0.38
ITGAL P20701 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984699 0.83 ALDH1A1 (0.47) ALDH1A1KDM4EKMT2A
SCHEMBL19984595 0.80 ALDH1A1 (0.44) ALDH1A1MAPTRAB9AKDM4EKMT2A
SCHEMBL21291444 0.76 HCRTR1 (0.51) ALDH1A1MAPK1KMT2A
SCHEMBL29360904 0.76 HCRTR1 (0.51) ALDH1A1MAPK1KMT2A
SCHEMBL19975023 0.73 FKBP1A (0.48) ALDH1A1MAPK1PKMRAB9AKMT2A
SCHEMBL31343689 0.71 MAPT (0.54) ALDH1A1MAPK1MAPTPKMRAB9A
SCHEMBL31343731 0.71 MAPT (0.54) ALDH1A1MAPK1MAPTPKMRAB9A
SCHEMBL18814405 0.71 MAPT (0.45) ALDH1A1HPGDMAPK1MAPTPKM
SCHEMBL7322642 0.70 LTA4H (0.46) ALDH1A1MAPTKMT2A
SCHEMBL2905551 0.69 SMN1; SMN2 (0.51) ALDH1A1MAPTNPC1PKMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053157-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2018-03-22 WO disclosed