SCHEMBL19984699

SCHEMBL19984699

COC(=O)C1CCCN1Sc1ccc(Br)cc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
AAK1 Q2M2I8 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
DRD2 P14416 1/20 0.35
CASP3 P42574 1/20 0.35
FPR2 P25090 1/20 0.34
SCN9A Q15858 1/20 0.34
CCR5 P51681 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
PEPD P12955 1/20 0.34
XPNPEP1 Q9NQW7 1/20 0.34
ALOX5 P09917 1/20 0.33
LTA4H P09960 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984595 0.97 ALDH1A1 (0.44) ALDH1A1AAK1HTTSMN1; SMN2CASP3
SCHEMBL19984522 0.85 ALDH1A1 (0.38) ALDH1A1AAK1SMN1; SMN2HCRTR1HCRTR2
SCHEMBL19984536 0.83 ALDH1A1 (0.45) ALDH1A1KDM4EKMT2A
SCHEMBL19984569 0.82 AAK1 (0.38) ALDH1A1AAK1HTTSMN1; SMN2KDM4E
SCHEMBL28305430 0.74 HCRTR1 (0.53) ALDH1A1SMN1; SMN2HCRTR1HCRTR2CASP3
SCHEMBL19984545 0.74 HCRTR1 (0.53) ALDH1A1SMN1; SMN2HCRTR1HCRTR2CASP3
SCHEMBL7322642 0.72 LTA4H (0.46) ALDH1A1SMN1; SMN2CASP3SCN9AMEN1
SCHEMBL19975403 0.71 HCRTR1 (0.50) ALDH1A1HCRTR1HCRTR2CASP3GAA
SCHEMBL20108320 0.68 CASP3 (0.41) ALDH1A1HCRTR1HCRTR2CASP3FPR2
SCHEMBL23119683 0.67 MAPT (0.53) ALDH1A1HTTSMN1; SMN2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053157-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2018-03-22 WO disclosed