SCHEMBL19984848

SCHEMBL19984848

COc1cccc(NC(=O)N[C@@H](CC(N)=O)c2nnc(-c3cnccn3)o2)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 2/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MITF O75030 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
THRB P10828 1/20 0.41
UTS2R Q9UKP6 1/20 0.40
RAF1 P04049 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATR Q13535 1/20 0.40
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CDK8 P49336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984978 0.86 TSHR (0.39) ALDH1A1SMN1; SMN2TSHRNPC1RAB9A
SCHEMBL19984843 0.78 NAMPT (0.49) ALDH1A1SMN1; SMN2TSHRNPC1RAB9A
SCHEMBL19866357 0.74 CD274 (0.52) MEN1KMT2A
SCHEMBL18078725 0.74 CD274 (0.52) MEN1KMT2A
SCHEMBL19984831 0.70 LRRK2 (0.35) ALDH1A1SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL14517931 0.69 KDM4E (0.74) ALDH1A1SMN1; SMN2TSHRNPC1RAB9A
SCHEMBL19973940 0.67 MAPK1 (0.33) MEN1KMT2A
SCHEMBL19984804 0.66 GAA (0.45) ALDH1A1SMN1; SMN2TSHRNPC1RAB9A
SCHEMBL19984850 0.65 HDAC6 (0.40) NPC1RAB9AGAAMAPTHTT
SCHEMBL19984811 0.65 KDM4E (0.43) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed