SCHEMBL19984978

SCHEMBL19984978

COc1cccc(NC(=O)N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)c2nnc(-c3cnccn3)o2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 3/20 0.39
MAPT P10636 3/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MITF O75030 1/20 0.38
SMN1; SMN2 Q16637 5/20 0.38
HTT P42858 3/20 0.38
PKM P14618 2/20 0.38
USP2 O75604 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 2/20 0.37
GAA P10253 1/20 0.37
CASR P41180 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984848 0.86 ALDH1A1 (0.43) TSHRALOX15HSD17B10MAPTNPC1
SCHEMBL19984980 0.77 PIEZO1 (0.38) MAPTNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL19984843 0.73 NAMPT (0.49) TSHRMAPTNPC1RAB9AALDH1A1
SCHEMBL14517931 0.65 KDM4E (0.74) TSHRTP53MAPTNPC1RAB9A
SCHEMBL30511404 0.62 ADAMTS4 (0.51) NPC1RAB9AALDH1A1SMN1; SMN2HTT
Benzene SCHEMBL11579880 0.61 THRB (0.71) TSHRTP53MAPTNPC1RAB9A
SCHEMBL30511402 0.61 ALDH1A1 (0.50) TSHRALOX15HSD17B10TP53MAPT
SCHEMBL14442613 0.61 TP53 (0.84) TSHRALOX15HSD17B10TP53MAPT
SCHEMBL19449478 0.60 THRB (0.72) TSHRTP53MAPTNPC1RAB9A
SCHEMBL4893387 0.59 TP53 (0.87) TSHRALOX15HSD17B10TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed