SCHEMBL19984831

SCHEMBL19984831

NC(=O)C[C@H](NC(=O)N1CCOCC1)c1nnc(-c2cnccn2)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.35
HDAC6 Q9UBN7 4/20 0.35
DYRK1A Q13627 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
GSK3B P49841 1/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
PKM P14618 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TNKS O95271 1/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
VNN1 O95497 2/20 0.32
ALDH1A1 P00352 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19984850 0.83 HDAC6 (0.40) LRRK2HDAC6DYRK1AHDAC1GSK3B
SCHEMBL19984975 0.76 TRHR (0.36) TNKSPARP1PARP2ALDH1A1
SCHEMBL19866357 0.74 CD274 (0.52) MEN1POLBKMT2A
SCHEMBL18078725 0.74 CD274 (0.52) MEN1POLBKMT2A
SCHEMBL19973940 0.72 MAPK1 (0.33) MEN1POLBKMT2A
SCHEMBL19973939 0.72 MAPK1 (0.33) MEN1POLBKMT2A
SCHEMBL19984824 0.71 HDAC6 (0.34) HDAC6CYP2C9CYP2C19
SCHEMBL19981151 0.67 SMN1; SMN2 (0.41) PKMSMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL19981270 0.66 BMP1 (0.40) LRRK2DYRK1AGSK3BPKMALDH1A1
SCHEMBL31153424 0.65 VNN1 (0.50) SMN1; SMN2VNN1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed