SCHEMBL19994485

SCHEMBL19994485

COC(=O)c1ccc(C(=O)c2ccco2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.71
SMN1; SMN2 Q16637 3/20 0.68
NPC1 O15118 3/20 0.68
RAB9A P51151 3/20 0.68
TP53 P04637 1/20 0.68
PSMD14 O00487 1/20 0.64
CACNA1B Q00975 1/20 0.64
APBA1 Q02410 1/20 0.64
MAOB P27338 1/20 0.62
MEN1 O00255 3/20 0.59
ALDH1A1 P00352 2/20 0.59
POLB P06746 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
THRB P10828 1/20 0.59
APEX1 P27695 1/20 0.59
RECQL P46063 1/20 0.59
HTT P42858 1/20 0.55
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13142806 0.83 KMT2A (0.62) KMT2ASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL23249749 0.82 KMT2A (0.66) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL30698159 0.81 KMT2A (0.69) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL363937 0.81
SCHEMBL2834430 0.81 RAB9A (1.00) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL10829218 0.81 KMT2A (0.61) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL10682751 0.80 ALDH1A1 (0.66) KMT2ASMN1; SMN2NPC1RAB9ATP53
Hydrochloric Acid SCHEMBL11748963 0.80 KMT2A (0.67) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL15056924 0.79 KMT2A (0.61) KMT2ASMN1; SMN2NPC1RAB9ATP53
SCHEMBL459833 0.78 MEN1 (0.68) KMT2ASMN1; SMN2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
CN-110234640-B Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2023-04-07 CN disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
EP-3515904-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS Centre Leon Berard (FR) 2019-07-31 EP disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CCAR2, MAPKAP1, BCOR KMT2A 3941/4885SMN1; SMN2 2392/4885NPC1 1805/4885
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS TMBIM6, BAX, MAPK14 KMT2A 3022/4885SMN1; SMN2 3155/4885NPC1 3255/4885
US-11384081-B2 Benzoimidazole derivatives as anticancer agents TMBIM6, BAX, MAPK14 KMT2A 3022/4885SMN1; SMN2 3155/4885NPC1 3255/4885
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents TMBIM6, BAX, BCL2 KMT2A 3028/4885SMN1; SMN2 3174/4885NPC1 3283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.