SCHEMBL19994736

SCHEMBL19994736

CN(C)c1ccc(-c2nc3cc(-c4ncccn4)ccc3[nH]2)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AURKA O14965 12/20 0.59
TCF4 P15884 1/20 0.54
CTNNB1 P35222 1/20 0.54
KIF11 P52732 1/20 0.50
MAPT P10636 3/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
GUSB P08236 1/20 0.48
RAB9A P51151 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
NOX1 Q9Y5S8 1/20 0.47
PARP1 P09874 1/20 0.43
CHEK2 O96017 1/20 0.43
SNCA P37840 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30343733 1.00 AURKA (0.59) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL13836671 0.87 TCF4 (0.64) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL19994448 0.83 ALDH1A1 (0.59) MAPTKDM4ENPC1GUSBRAB9A
SCHEMBL13974405 0.82 TCF4 (0.70) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL31005274 0.80 TCF4 (0.59) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL17370980 0.80 TCF4 (0.59) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL31005272 0.80 TCF4 (0.59) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL2554510 0.80 NPC1 (0.58) AURKAMAPTKDM4ENPC1GUSB
SCHEMBL1663529 0.79 TCF4 (0.58) AURKATCF4CTNNB1KIF11MAPT
SCHEMBL29506637 0.79 TCF4 (0.79) AURKATCF4CTNNB1KIF11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed
CN-110234640-B Benzimidazole derivatives as anticancer agents 利昂贝拉尔中心 2023-04-07 CN disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents CENTRE LEON BERARD (FR) 2022-11-03 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-11384081-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2022-07-12 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2021-09-23 US disclosed
EP-3515904-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS Centre Leon Berard (FR) 2019-07-31 EP disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CCAR2, MAPKAP1, BCOR AURKA 1394/4885TCF4 3369/4885CTNNB1 1287/4885
US-20210292328-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS TMBIM6, BAX, MAPK14 AURKA 347/4885TCF4 2690/4885CTNNB1 1908/4885
US-11384081-B2 Benzoimidazole derivatives as anticancer agents TMBIM6, BAX, MAPK14 AURKA 347/4885TCF4 2690/4885CTNNB1 1908/4885
US-20220348587-A1 Benzoimidazole Derivatives As Anticancer Agents TMBIM6, BAX, BCL2 AURKA 376/4885TCF4 2717/4885CTNNB1 1960/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.