SCHEMBL20000528

SCHEMBL20000528

CC(F)(F)COc1ncnc(N)c1F

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACACB O00763 16/20 0.36
MBOAT4 Q96T53 2/20 0.34
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
NUDT1 P36639 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20000527 0.85 MAP3K7 (0.40) ACACBMBOAT4PI4KAPI4K2BPI4K2A
SCHEMBL38661744 0.74 PDPK1 (0.37) PI4KAPI4K2BPI4K2API4KB
SCHEMBL16190524 0.73 ACACB (0.49) ACACB
SCHEMBL15741407 0.67
SCHEMBL16822073 0.67 CYP2C9 (0.38) MBOAT4NUDT1
SCHEMBL19004852 0.67 CA2 (0.44) MBOAT4NUDT1
SCHEMBL18809713 0.66
SCHEMBL24714020 0.66 PI4KA (0.36) PI4KAPI4K2BPI4K2API4KB
SCHEMBL10569355 0.66 ALDH1A1 (0.45) MBOAT4NUDT1
SCHEMBL1440438 0.65 CA2 (0.40) PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997024-B1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2018-03-28 EP disclosed