SCHEMBL20002322

SCHEMBL20002322

O=C(N1CCOCC1)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.60
AKR1C3 P42330 2/20 0.52
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RORC P51449 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
EPHX2 P34913 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
KCNH2 Q12809 1/20 0.43
AKT1 P31749 1/20 0.42
PIK3CA P42336 1/20 0.42
PHGDH O43175 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002563 0.87 EPHX2 (0.45) PKMMEN1KMT2AL3MBTL1EPHX2
SCHEMBL20003003 0.87 EPHX2 (0.45) PKMRORCL3MBTL1EPHX2HTR2A
SCHEMBL20002321 0.85 CCR5 (0.46) PKMRORCEPHX2
SCHEMBL20002221 0.85 RORC (0.45) PKMRORCL3MBTL1EPHX2SMN1; SMN2
SCHEMBL20003053 0.85 CCR5 (0.46) PKMRORCEPHX2
SCHEMBL20002459 0.85 RORC (0.51) PKMAKR1C3RORCEPHX2HTR2A
SCHEMBL20003234 0.84 HTR2A (0.45) PKMRORCL3MBTL1EPHX2HTR2A
SCHEMBL20003027 0.84 EPHX2 (0.43) PKMRORCL3MBTL1EPHX2HTR2A
SCHEMBL20003031 0.84 EPHX2 (0.44) PKMRORCL3MBTL1EPHX2HTR2A
SCHEMBL20003035 0.83 HTR2A (0.44) PKMRORCL3MBTL1EPHX2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed