SCHEMBL20003035

SCHEMBL20003035

CN(C)C1CCN(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.44
HTR2C P28335 3/20 0.44
L3MBTL3 Q96JM7 2/20 0.44
RORC P51449 2/20 0.44
TSHR P16473 1/20 0.42
EPHX2 P34913 1/20 0.42
KCNH2 Q12809 2/20 0.41
MCHR1 Q99705 1/20 0.41
PKM P14618 1/20 0.40
CCR5 P51681 1/20 0.39
DRD2 P14416 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
GPR6 P46095 1/20 0.38
USP5 P45974 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003053 0.85 CCR5 (0.46) RORCEPHX2PKMCCR5GPR6
SCHEMBL20002221 0.85 RORC (0.45) HTR2AHTR2CRORCEPHX2KCNH2
SCHEMBL20002321 0.85 CCR5 (0.46) RORCEPHX2PKMCCR5GPR6
SCHEMBL20002563 0.85 EPHX2 (0.45) HTR2AHTR2CEPHX2KCNH2PKM
SCHEMBL20003003 0.85 EPHX2 (0.45) HTR2AHTR2CRORCEPHX2KCNH2
SCHEMBL20002459 0.83 RORC (0.51) HTR2AHTR2CRORCEPHX2KCNH2
SCHEMBL20002322 0.83 PKM (0.60) HTR2AHTR2CRORCEPHX2KCNH2
SCHEMBL20002346 0.82 RORC (0.50) HTR2AHTR2CRORCEPHX2KCNH2
SCHEMBL20003234 0.82 HTR2A (0.45) HTR2AHTR2CRORCTSHREPHX2
SCHEMBL20003027 0.82 EPHX2 (0.43) HTR2AHTR2CRORCEPHX2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed