SCHEMBL20002459

SCHEMBL20002459

O=C(O)C1CCN(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 11/20 0.51
MAPT P10636 1/20 0.49
NOTUM Q6P988 1/20 0.46
HTR2A P28223 2/20 0.46
HTR2C P28335 1/20 0.46
KCNH2 Q12809 1/20 0.46
EPHX2 P34913 1/20 0.43
DRD2 P14416 1/20 0.42
HSD11B1 P28845 1/20 0.42
AKR1C3 P42330 1/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002498 0.88 RORC (0.49) RORCMAPTHTR2AHTR2CKCNH2
SCHEMBL20002563 0.87 EPHX2 (0.45) MAPTHTR2AHTR2CKCNH2EPHX2
SCHEMBL20003003 0.87 EPHX2 (0.45) RORCMAPTHTR2AHTR2CKCNH2
SCHEMBL20002942 0.86 RORC (0.45) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002321 0.85 CCR5 (0.46) RORCEPHX2PKM
SCHEMBL20003053 0.85 CCR5 (0.46) RORCEPHX2PKM
SCHEMBL20002322 0.85 PKM (0.60) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002221 0.85 RORC (0.45) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002933 0.84 RORC (0.46) RORCMAPTHTR2AHTR2CKCNH2
SCHEMBL20003234 0.84 HTR2A (0.45) RORCMAPTHTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed