SCHEMBL20002221

SCHEMBL20002221

CN1CCN(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.45
PKM P14618 2/20 0.44
EPHX2 P34913 1/20 0.43
HTR2A P28223 5/20 0.43
HTR2C P28335 4/20 0.43
KCNH2 Q12809 3/20 0.43
MMP1 P03956 1/20 0.43
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
MMP9 P14780 1/20 0.43
MMP13 P45452 1/20 0.43
DRD2 P14416 2/20 0.42
ALOX5 P09917 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CCR5 P51681 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002321 0.90 CCR5 (0.46) RORCPKMEPHX2CCR5
SCHEMBL20003053 0.90 CCR5 (0.46) RORCPKMEPHX2CCR5
SCHEMBL20002907 0.88 RORC (0.42) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20002563 0.87 EPHX2 (0.45) PKMEPHX2HTR2AHTR2CKCNH2
SCHEMBL20003003 0.87 EPHX2 (0.45) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20003234 0.86 HTR2A (0.45) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20003035 0.85 HTR2A (0.44) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20002322 0.85 PKM (0.60) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20002459 0.85 RORC (0.51) RORCPKMEPHX2HTR2AHTR2C
SCHEMBL20002346 0.84 RORC (0.50) RORCPKMEPHX2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed