SCHEMBL20002346

SCHEMBL20002346

CC1(O)CCN(C(=O)N2CC[C@H](S(=O)(=O)c3ccc(F)cc3)C2)CC1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 17/20 0.50
EPHX2 P34913 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
KCNH2 Q12809 1/20 0.41
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002899 0.88 RORC (0.44) RORC
SCHEMBL20002526 0.86 RORC (0.53) RORCEPHX2
SCHEMBL20003007 0.86 RORC (0.44) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002321 0.84 CCR5 (0.46) RORCEPHX2PKM
SCHEMBL20002221 0.84 RORC (0.45) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20003053 0.84 CCR5 (0.46) RORCEPHX2PKM
SCHEMBL20003003 0.84 EPHX2 (0.45) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002563 0.84 EPHX2 (0.45) EPHX2HTR2AHTR2CKCNH2PKM
SCHEMBL20003035 0.82 HTR2A (0.44) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002459 0.82 RORC (0.51) RORCEPHX2HTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed