SCHEMBL20002429

SCHEMBL20002429

CC(=O)N1CCN(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)C[C@H]1CO

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.41
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
CA9 Q16790 2/20 0.33
OPRK1 P41145 1/20 0.33
TRPC6 Q9Y210 4/20 0.33
TACR1 P25103 1/20 0.32
HSD11B1 P28845 3/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002280 0.85 TACR1 (0.40) RORCTACR1HSD11B1
SCHEMBL20002167 0.80 KDM1A (0.40) RORCSMN1; SMN2
SCHEMBL20002664 0.77 TSHR (0.41) HSD11B1SMN1; SMN2
SCHEMBL20002990 0.77 RORC (0.40) RORCCA1CA2CA4CA9
SCHEMBL20002669 0.76 NOTUM (0.45) RORCHSD11B1SMN1; SMN2
SCHEMBL20002958 0.76 NOTUM (0.48) RORCHSD11B1SMN1; SMN2
SCHEMBL20002957 0.76 NOTUM (0.48) RORCHSD11B1SMN1; SMN2
SCHEMBL20002969 0.76 NOTUM (0.45) RORCHSD11B1SMN1; SMN2
SCHEMBL20003049 0.76 AKR1C3 (0.51) HSD11B1SMN1; SMN2
SCHEMBL20003029 0.75 RORC (0.41) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed