SCHEMBL20002167

SCHEMBL20002167

CN1CCN(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.40
MAOB P27338 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 1/20 0.40
EPHX2 P34913 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
CYP2D6 P10635 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
AKR1C3 P42330 1/20 0.36
RORC P51449 1/20 0.36
PKM P14618 1/20 0.36
FAAH O00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002280 0.90 TACR1 (0.40) AKR1C3RORCPKM
SCHEMBL20002664 0.87 TSHR (0.41) SMN1; SMN2NPC1LMNARAB9AAKR1C3
SCHEMBL20003049 0.85 AKR1C3 (0.51) SMN1; SMN2HTTEPHX2ALDH1A1NPC1
SCHEMBL20002669 0.85 NOTUM (0.45) SMN1; SMN2ALDH1A1LMNARAB9AAKR1C3
SCHEMBL20002969 0.85 NOTUM (0.45) SMN1; SMN2ALDH1A1LMNARAB9AAKR1C3
SCHEMBL20003029 0.85 RORC (0.41) KDM1ARORC
SCHEMBL20002631 0.84 HSD11B1 (0.33) SMN1; SMN2ALDH1A1NPC1LMNARAB9A
SCHEMBL20002564 0.84 NAMPT (0.41) SMN1; SMN2ALDH1A1LMNA
SCHEMBL20002957 0.83 NOTUM (0.48) SMN1; SMN2EPHX2ALDH1A1LMNAAKR1C3
SCHEMBL20002958 0.83 NOTUM (0.48) SMN1; SMN2EPHX2ALDH1A1LMNAAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed