SCHEMBL20002957

SCHEMBL20002957

O=C(O)[C@@H]1CCN(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.48
MAPT P10636 1/20 0.43
HSD11B1 P28845 7/20 0.39
RORC P51449 6/20 0.38
LMNA P02545 2/20 0.37
KMT2A Q03164 1/20 0.37
AKR1C3 P42330 1/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EPHX2 P34913 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002958 1.00 NOTUM (0.48) NOTUMMAPTHSD11B1RORCLMNA
SCHEMBL20002669 0.95 NOTUM (0.45) NOTUMMAPTHSD11B1RORCLMNA
SCHEMBL20002969 0.95 NOTUM (0.45) NOTUMMAPTHSD11B1RORCLMNA
SCHEMBL20002341 0.94 MAPT (0.48) NOTUMMAPTRORCKMT2AALDH1A1
SCHEMBL20002250 0.94 MAPT (0.48) NOTUMMAPTRORCKMT2AALDH1A1
SCHEMBL20002751 0.85 NOTUM (0.42) NOTUMMAPTRORC
SCHEMBL20002773 0.85 RORC (0.44) NOTUMMAPTHSD11B1RORCLMNA
SCHEMBL20003049 0.83 AKR1C3 (0.51) HSD11B1LMNAKMT2AAKR1C3ALDH1A1
SCHEMBL20002280 0.83 TACR1 (0.40) HSD11B1RORCAKR1C3
SCHEMBL20002167 0.83 KDM1A (0.40) RORCLMNAAKR1C3ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed