SCHEMBL20003049

SCHEMBL20003049

O=C(N1CCOCC1)N1CCC([S+]([O-])c2ccc(F)cc2)C1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.51
PKM P14618 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.42
PHGDH O43175 1/20 0.41
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
HSD11B1 P28845 1/20 0.40
FKBP1A P62942 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
EPHX2 P34913 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002669 0.85 NOTUM (0.45) AKR1C3SMN1; SMN2LMNAHSD11B1KMT2A
SCHEMBL20002280 0.85 TACR1 (0.40) AKR1C3PKMHSD11B1
SCHEMBL20002167 0.85 KDM1A (0.40) AKR1C3PKMSMN1; SMN2LMNAHTT
SCHEMBL20002969 0.85 NOTUM (0.45) AKR1C3SMN1; SMN2LMNAHSD11B1KMT2A
SCHEMBL20002664 0.84 TSHR (0.41) AKR1C3PKMSMN1; SMN2LMNAHSD11B1
SCHEMBL20002631 0.84 HSD11B1 (0.33) AKR1C3PKMSMN1; SMN2LMNAHSD11B1
SCHEMBL20002400 0.84 TACR3 (0.42) SMN1; SMN2HTTHSD11B1MEN1KMT2A
SCHEMBL20002957 0.83 NOTUM (0.48) AKR1C3SMN1; SMN2LMNAHSD11B1KMT2A
SCHEMBL20002958 0.83 NOTUM (0.48) AKR1C3SMN1; SMN2LMNAHSD11B1KMT2A
SCHEMBL20003029 0.82 RORC (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed