SCHEMBL20002495

SCHEMBL20002495

O=C(CO)N1CC[C@@H](C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.40
NR1I2 O75469 2/20 0.40
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.38
ALOX12 P18054 1/20 0.38
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
HSD11B1 P28845 1/20 0.36
CYP46A1 Q9Y6A2 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002943 0.87 RORC (0.47) RORCNR1I2MAPTPKMALOX12
SCHEMBL20002698 0.85 HSD11B1 (0.47) RORCKMT2AALDH1A1SMN1; SMN2HSD11B1
SCHEMBL20002706 0.85 HSD11B1 (0.47) RORCKMT2AALDH1A1SMN1; SMN2HSD11B1
SCHEMBL20002564 0.83 NAMPT (0.41) KMT2AALDH1A1SMN1; SMN2GAAHSD11B1
SCHEMBL20002286 0.83 TACR1 (0.45) RORCNR1I2
SCHEMBL20002987 0.82 TACR3 (0.49) RORCNR1I2MAPTPKMALOX12
SCHEMBL20002685 0.81 HSD11B1 (0.41) RORCMAPTPKMALOX12ALDH1A1
SCHEMBL20002751 0.81 NOTUM (0.42) RORCMAPTL3MBTL1
SCHEMBL20002854 0.81 RORC (0.42) RORCMAPTPKMALOX12KMT2A
SCHEMBL20002400 0.81 TACR3 (0.42) RORCMAPTKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed