SCHEMBL20002690

SCHEMBL20002690

N#Cc1ccc(CC(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 2/20 0.50
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
KCNH2 Q12809 1/20 0.49
CNR1 P21554 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
ALDH1A1 P00352 1/20 0.48
RORC P51449 4/20 0.46
KDM1A O60341 3/20 0.45
MLNR O43193 3/20 0.42
AKT1 P31749 1/20 0.42
PIK3CA P42336 1/20 0.42
POLB P06746 1/20 0.42
EPHX2 P34913 1/20 0.41
NSD2 O96028 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002837 0.84 RORC (0.49) HTR2AHTR2CKCNH2SMN1; SMN2ALDH1A1
SCHEMBL20003002 0.78 TSHR (0.48) SMN1; SMN2ALDH1A1RORC
SCHEMBL19702674 0.77 SMN1; SMN2 (0.54) PRKAA2SMN1; SMN2ALDH1A1POLB
SCHEMBL7030971 0.76 HTR2A (0.73) PRKAA2HTR2AHTR2CKCNH2
SCHEMBL12385821 0.74 ALDH1A1 (0.59) CNR1SMN1; SMN2ALDH1A1KDM1AMLNR
SCHEMBL20002968 0.74 RORC (0.48) PRKAA2HTR2AHTR2CKCNH2RORC
SCHEMBL16632052 0.74 HTR2A (0.49) PRKAA2HTR2AHTR2CKCNH2KDM1A
SCHEMBL14413535 0.74 EPHX2 (0.47) HTR2AHTR2CKCNH2RORCPOLB
SCHEMBL6585537 0.74 HTR2A (0.73) PRKAA2HTR2AHTR2CKCNH2SMN1; SMN2
SCHEMBL15231711 0.73 HTR2A (0.48) PRKAA2HTR2AHTR2CKCNH2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed