SCHEMBL20002823

SCHEMBL20002823

CC12CCC(C(=O)N3CCC(Sc4ccc(F)cc4)C3)(CC1)CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.38
KMT2A Q03164 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ATM Q13315 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.34
HSD11B1 P28845 7/20 0.33
GFER P55789 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003154 0.89 RORC (0.39) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20003220 0.86 RORC (0.41) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20003191 0.85 RORC (0.41) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20002430 0.79 RORC (0.44) CCR5KMT2AHDAC3HDAC1HDAC2
SCHEMBL20002294 0.78 PTPN11 (0.36) CCR5KMT2AGRIN1GRIN2BDDB1
SCHEMBL20003080 0.78 GRIN1 (0.35) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20003055 0.77 RORC (0.42) KMT2ANPC1RAB9AALDH1A1TSHR
SCHEMBL20002375 0.77 RORC (0.41) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20002612 0.77 RORC (0.36) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20002936 0.77 CCR5 (0.46) CCR5KMT2AGRIN1GRIN2BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed