SCHEMBL20003080

SCHEMBL20003080

O=C(N1CCC(Sc2ccc(F)cc2)C1)C1(O)CCSCC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ATM Q13315 1/20 0.34
FASN P49327 2/20 0.34
CCR5 P51681 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 1/20 0.33
PKM P14618 1/20 0.33
HSD11B1 P28845 4/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
RIPK1 Q13546 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPT P10636 1/20 0.32
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003154 0.79 RORC (0.39) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20002823 0.78 CCR5 (0.38) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20003191 0.77 RORC (0.41) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20002375 0.76 RORC (0.41) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20003220 0.76 RORC (0.41) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20003026 0.73 RORC (0.47) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20002430 0.73 RORC (0.44) CCR5KMT2ARORC
SCHEMBL20003152 0.73 RAB9A (0.34) GRIN1GRIN2BNPC1RAB9AATM
SCHEMBL20002294 0.72 PTPN11 (0.36) GRIN1GRIN2BCCR5KMT2ADDB1
SCHEMBL20002719 0.72 HSD11B1 (0.48) ALDH1A1KMT2AHSD11B1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed