SCHEMBL20002612

SCHEMBL20002612

CC1(C(=O)O)CCN(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.36
CCR5 P51681 1/20 0.35
CACNA1B Q00975 2/20 0.35
KMT2A Q03164 1/20 0.35
NOTUM Q6P988 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
KCNK3 O14649 1/20 0.34
RIPK1 Q13546 1/20 0.33
DPP4 P27487 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002294 0.87 PTPN11 (0.36) RORCCCR5CACNA1BKMT2ADDB1
SCHEMBL20002879 0.83 NPC1 (0.44) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20002297 0.82 NOTUM (0.47) RORCCCR5KMT2ANOTUMGRIN1
SCHEMBL20002936 0.82 CCR5 (0.46) CCR5KMT2AGRIN1GRIN2BDPP4
SCHEMBL20002407 0.82 SMN1; SMN2 (0.41) CCR5KMT2AGRIN1GRIN2BNPC1
SCHEMBL20003024 0.80 NOTUM (0.44) CCR5CACNA1BKMT2ANOTUMGRIN1
SCHEMBL20003154 0.78 RORC (0.39) RORCCCR5CACNA1BKMT2ANOTUM
SCHEMBL20002823 0.77 CCR5 (0.38) CCR5KMT2ADDB1CRBNGRIN1
SCHEMBL20003191 0.76 RORC (0.41) RORCCCR5CACNA1BKMT2ANOTUM
SCHEMBL4097076 0.73 CCR5 (0.42) CCR5CACNA1BKMT2ANOTUMDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed