SCHEMBL20002294

SCHEMBL20002294

CC1(N)CCN(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 3/20 0.36
CCR5 P51681 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
RORC P51449 6/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
MAPK1 P28482 1/20 0.34
RIPK1 Q13546 1/20 0.34
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002612 0.87 RORC (0.36) CCR5KMT2ADDB1CRBNRORC
SCHEMBL20002879 0.84 NPC1 (0.44) CCR5KMT2ACHRM2GRIN1GRIN2B
SCHEMBL20002936 0.83 CCR5 (0.46) CCR5KMT2AGRIN1GRIN2BDPP4
SCHEMBL20002407 0.83 SMN1; SMN2 (0.41) CCR5KMT2AGRIN1GRIN2BRIPK1
SCHEMBL20002297 0.81 NOTUM (0.47) CCR5KMT2ARORCGRIN1GRIN2B
SCHEMBL20003024 0.78 NOTUM (0.44) CCR5KMT2AGRIN1GRIN2BRIPK1
SCHEMBL20002823 0.78 CCR5 (0.38) CCR5KMT2ADDB1CRBNGRIN1
SCHEMBL20002375 0.76 RORC (0.41) CCR5KMT2ARORCGRIN1GRIN2B
SCHEMBL20002430 0.76 RORC (0.44) CCR5KMT2ARORCDPP4DPP8
SCHEMBL20003154 0.74 RORC (0.39) CCR5KMT2ARORCGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed