SCHEMBL20003153

SCHEMBL20003153

CC1(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CC[S+]([O-])CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.41
EPHX2 P34913 1/20 0.40
PSEN1 P49768 2/20 0.39
PSEN2 P49810 2/20 0.39
APH1B Q8WW43 2/20 0.39
NCSTN Q92542 2/20 0.39
APH1A Q96BI3 2/20 0.39
PSENEN Q9NZ42 2/20 0.39
HTR2A P28223 3/20 0.39
HTR2C P28335 2/20 0.39
KCNH2 Q12809 2/20 0.39
DRD2 P14416 1/20 0.36
GPR6 P46095 1/20 0.35
CCR5 P51681 1/20 0.35
FASN P49327 2/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002406 0.87 RORC (0.42) RORCEPHX2PSEN1PSEN2APH1B
SCHEMBL20002497 0.86 RORC (0.44) RORCPSEN1PSEN2APH1BNCSTN
SCHEMBL20002684 0.80 L3MBTL1 (0.47) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002866 0.77 RORC (0.49) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002346 0.76 RORC (0.50) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002978 0.76 RORC (0.42) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002921 0.76 RORC (0.44) RORCGPR6CCR5
SCHEMBL20002899 0.76 RORC (0.44) RORC
SCHEMBL20003156 0.76 L3MBTL1 (0.43) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002869 0.75 RORC (0.44) RORCEPHX2HTR2AHTR2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed