SCHEMBL20002902

SCHEMBL20002902

CC(=O)N1CCN(C(=O)N2CC[C@H]([S+]([O-])c3ccc(Oc4ccccc4)cc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MAPK1 P28482 1/20 0.47
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RORC P51449 1/20 0.41
HTT P42858 1/20 0.40
BTK Q06187 2/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EPHX2 P34913 1/20 0.37
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002280 0.84 TACR1 (0.40) RORC
SCHEMBL20149113 0.76 RORC (0.39) ALDH1A1RORCMEN1KMT2A
SCHEMBL20002167 0.74 KDM1A (0.40) ALDH1A1MMP9NPC1RAB9ALMNA
SCHEMBL20002664 0.74 TSHR (0.41) MAPK1NPC1RAB9ALMNASMN1; SMN2
SCHEMBL20002969 0.72 NOTUM (0.45) ALDH1A1RAB9ALMNASMN1; SMN2RORC
SCHEMBL20002669 0.72 NOTUM (0.45) ALDH1A1RAB9ALMNASMN1; SMN2RORC
SCHEMBL20002286 0.71 TACR1 (0.45) RORC
SCHEMBL20002429 0.70 RORC (0.41) SMN1; SMN2RORC
SCHEMBL20002958 0.70 NOTUM (0.48) ALDH1A1LMNASMN1; SMN2RORCKMT2A
SCHEMBL20003049 0.70 AKR1C3 (0.51) ALDH1A1NPC1LMNASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed