SCHEMBL20002460

SCHEMBL20002460

CC(=O)NC1(C(=O)N2CCC(S(=O)(=O)c3ccc(F)cc3)C2)CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.55
MMP13 P45452 6/20 0.41
MMP1 P03956 4/20 0.41
EPHX2 P34913 1/20 0.39
MMP2 P08253 3/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP14 P50281 1/20 0.39
AKT1 P31749 1/20 0.37
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
GPR6 P46095 1/20 0.37
PKM P14618 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002922 0.89 RORC (0.46) RORCEPHX2GPR6
SCHEMBL20002566 0.79 RORC (0.46) RORCMMP13MMP1MMP2MMP3
SCHEMBL20002322 0.76 PKM (0.60) RORCEPHX2AKT1PIK3CAPKM
SCHEMBL20002497 0.76 RORC (0.44) RORCGPR6
SCHEMBL20002921 0.75 RORC (0.44) RORCGPR6
SCHEMBL20002406 0.75 RORC (0.42) RORCEPHX2HTR2AHTR2CKCNH2
SCHEMBL20002866 0.74 RORC (0.49) RORCEPHX2GPR6HTR2AHTR2C
SCHEMBL13890294 0.73 EPHX2 (0.50) EPHX2GPR6PKMHTR2AHTR2C
SCHEMBL20003153 0.73 RORC (0.41) RORCEPHX2GPR6HTR2AHTR2C
SCHEMBL20003009 0.73 RORC (0.54) RORCEPHX2GPR6HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed